Microwave-assisted synthesis of α-aminophosphonates with sterically demanding α-aryl substituents
نویسندگان
چکیده
منابع مشابه
The synthesis of α-aryl-α-aminophosphonates and α-aryl-α-aminophosphine oxides by the microwave-assisted Pudovik reaction
A family of α-aryl-α-aminophosphonates and α-aryl-α-aminophosphine oxides was synthesized by the microwave-assisted solvent-free addition of dialkyl phosphites and diphenylphosphine oxide, respectively, to imines formed from benzaldehyde derivatives and primary amines. After optimization, the reactivity was mapped, and the fine mechanism was evaluated by DFT calculations. Two α-aminophosphonate...
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ژورنال
عنوان ژورنال: Synthetic Communications
سال: 2020
ISSN: 0039-7911,1532-2432
DOI: 10.1080/00397911.2019.1679186